Universität zu Köln

Humpert, Swen ORCID: 0000-0002-1995-0714, Omrane, Mohamed A., Urusova, Elizaveta A., Gremer, Lothar ORCID: 0000-0001-7065-5027, Willbold, Dieter ORCID: 0000-0002-0065-7366, Endepols, Heike, Krasikova, Raisa N., Neumaier, Bernd ORCID: 0000-0001-5425-3116 and Zlatopolskiy, Boris D. (2021). Rapid F-18-labeling via Pd-catalyzed S-arylation in aqueous medium. Chem. Commun., 57 (29). S. 3547 - 3551. CAMBRIDGE: ROYAL SOC CHEMISTRY. ISSN 1364-548X

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Abstract

We report radiolabeling of thiol-containing substrates via Pd-catalyzed S-arylation with 2-[F-18]fluoro-5-iodopyridine, which is readily accessible using the minimalist radiofluorination method. The practicality of the procedure was confirmed by preparation of a novel PSMA-specific PET-tracer as well as labeling of glutathione, A beta oligomer-binding RD2 peptide, bovine serum albumin and PSMA I&S.

Item Type:	Journal Article
Creators:	Creators Email ORCID ORCID Put Code Humpert, Swen UNSPECIFIED orcid.org/0000-0002-1995-0714 UNSPECIFIED Omrane, Mohamed A. UNSPECIFIED UNSPECIFIED UNSPECIFIED Urusova, Elizaveta A. UNSPECIFIED UNSPECIFIED UNSPECIFIED Gremer, Lothar UNSPECIFIED orcid.org/0000-0001-7065-5027 UNSPECIFIED Willbold, Dieter UNSPECIFIED orcid.org/0000-0002-0065-7366 UNSPECIFIED Endepols, Heike UNSPECIFIED UNSPECIFIED UNSPECIFIED Krasikova, Raisa N. UNSPECIFIED UNSPECIFIED UNSPECIFIED Neumaier, Bernd UNSPECIFIED orcid.org/0000-0001-5425-3116 UNSPECIFIED Zlatopolskiy, Boris D. UNSPECIFIED UNSPECIFIED UNSPECIFIED
URN:	urn:nbn:de:hbz:38-596453
DOI:	10.1039/d1cc00745a
Journal or Publication Title:	Chem. Commun.
Volume:	57
Number:	29
Page Range:	S. 3547 - 3551
Date:	2021
Publisher:	ROYAL SOC CHEMISTRY
Place of Publication:	CAMBRIDGE
ISSN:	1364-548X
Language:	English
Faculty:	Unspecified
Divisions:	Unspecified
Subjects:	no entry
Uncontrolled Keywords:	Keywords Language Chemistry, Multidisciplinary Multiple languages
URI:	http://kups.ub.uni-koeln.de/id/eprint/59645